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IDH1

3 drugs

Isocitrate Dehydrogenase 1

Predictive biomarker for patient selection in 5 indications

Understanding IDH1

What it means: IDH1 mutations produce 2-hydroxyglutarate, an oncometabolite that blocks cell differentiation. Found in AML and gliomas.
Why it matters: IDH1 inhibitors (ivosidenib) induce differentiation and show responses in IDH1-mutant AML and cholangiocarcinoma.
Testing: Tested via NGS or PCR. R132 mutations are most common. Also detectable via immunohistochemistry.
3
Approved Drugs
5
Indications
2
Companies
Search IDH1 Clinical Trials

Search recruiting trials on ClinicalTrials.gov

Drugs Targeting IDH1

Drug Company Therapeutic Area
REZLIDHIA RIGEL PHARMS Oncology
TIBSOVO SERVIER Oncology
VORANIGO SERVIER Oncology

Companies with IDH1 Drugs