TheraRadar
Data updated: May 26, 2026

BENZNIDAZOLE

Trial Activity: Declining 2 active trials
Orphan Drug Priority Review Accelerated Approval
Infectious Disease Approved 2017-08-29

BENZNIDAZOLE is indicated for the treatment of Chagas Disease; American Trypanosomiasis.

Source: FDA Label • CHEMO RESEARCH SL

How BENZNIDAZOLE Works

Benznidazole is a nitroimidazole antimicrobial drug that targets the *Trypanosoma cruzi* parasite. Its antimicrobial activity leads to a reduction in the parasite load, which is clinically manifested by a decrease in and eventual disappearance of specific IgG antibodies produced by the host against *T. cruzi* antigens.

Development Insights

Hospital Universitari Vall d'Hebron Research Institute conducting 2 trials (18%)
3 indications explored (Focused)
chagas disease (10 trials)
trypanosoma cruzi infection (2 trials)
safety issues (1 trials)
1
Indication
--
Phase 3 Trials
1
Priority Reviews
8
Years on Market

Details

Status
Prescription
First Approved
2017-08-29
Routes
ORAL
Dosage Forms
TABLET

Companies

Active Ingredient: BENZNIDAZOLE

BENZNIDAZOLE Approval History

2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
6 FDA actions from 2017 to 2021
Dec 2021 SUPPL
Label · Labeling
Nov 2019 SUPPL
Label · Labeling
Aug 2017 ORIGINAL Priority
New Drug · Type 1 - New Molecular Entity

What BENZNIDAZOLE Treats

2 indications

BENZNIDAZOLE is approved for 2 conditions since its original approval in 2017. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Chagas Disease
  • American Trypanosomiasis
Source: FDA Label

BENZNIDAZOLE Competitive Set

Pro

Three rings of competition based on shared molecular targets and treated indications.

Indication competitors

1

Same indication, different mechanism — what else might this patient receive?

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to BENZNIDAZOLE

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

LAMPIT
NIFURTIMOX
2 shared
Bayer
Shared indications:
Chagas DiseaseAmerican Trypanosomiasis
📋

Clinical Trial Registry

11 trials
Trial Sponsor ID Phase Status Title
NCT04024163 LPRI747-301 Ph 3 active not recruiting Prospective Study of Benznidazole for Chagas' Disease Children With Chronic Indeterminate Chagas Disease
NCT05523596 ICM003 Ph 1 completed A Phase 1 Study of the Safety and Tolerability of ICM20 in Adults
NCT03672487 BETTY results posted R01HD095857 Ph 3 completed Short-course Benznidazole Treatment to Reduce Trypanosoma Cruzi Parasitic Load in Women of Reproductive Age
NCT06632600 CLXE408B12201 Ph 2 recruiting A Study of Efficacy, Safety, Tolerability of LXE408 in Participants With Chronic Chagas Disease.
NCT03981523 TESEO 743474 U01AI129783 Ph 2 completed New Therapies and Biomarkers for Chagas Infection
NCT03191162 MULTIBENZ 2016-003789-21 Ph 2 completed Evaluation of Different Benznidazole Regimens for the Treatment of Chronic Chagas Disease.
NCT03892213 DNDi-CH-E1224-002 Ph 1 completed Pharmacokinetic Drug-Drug Interaction Study
NCT01377480 STOP CHAGAS results posted P05267 MK-5592-055 Ph 2 completed A Study of the Use of Oral Posaconazole (POS) in the Treatment of Asymptomatic Chronic Chagas Disease (P05267)
NCT01678599 PCR MSF/DNDi-CD-PCR-01 Ph 4 completed Optimization of PCR Technique to Assess Parasitological Response for Patients With Chronic Chagas Disease
NCT01755403 CINEBENZ CINEBENZ Ph 4 completed Population Pharmacokinetics in Benznidazole-treated Adults With Chronic With Chagas Disease
NCT01162967 CHAGASAZOL CHAGASAZOL01 Ph 2 completed Clinical Trial For The Treatment Of Chronic Chagas Disease With Posaconazole And Benznidazole
🔬

Active Pipeline

Pro

Ongoing clinical trials by development phase

Loading...

Key Completed Trials

Pro

Completed studies with published results, ranked by significance

Loading...
📊

Trial Timeline

Full development history with FDA approval milestones

|
Loading...
Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

BENZNIDAZOLE FDA Label Details

Indications & Usage

FDA Label (PDF)

BENZNIDAZOLE is indicated for the treatment of Chagas Disease; American Trypanosomiasis.

Track BENZNIDAZOLE with TheraRadar Pro

Watchlist alerts, full database access, CSV exports across 14,000+ drugs.

Upgrade to Pro

Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment