TheraRadar
Data updated: May 26, 2026

MILOPHENE (clomiphene citrate)

Trial Activity: Mature 5 active trials
Women's Health Approved 1988-12-20

MILOPHENE is indicated for the treatment of Ovulatory Dysfunction; Polycystic Ovary Syndrome; Amenorrhea-Galactorrhea Syndrome; Psychogenic Amenorrhea; Secondary Amenorrhea.

Source: FDA Label • GRANATA BIO CORP

Development Insights

Ain Shams University conducting 4 trials (11%)
34 indications explored (Broad Platform)
polycystic ovary syndrome (10 trials)
infertility (6 trials)
unexplained infertility (3 trials)
1
Indication
--
Phase 3 Trials
37
Years on Market

Details

Status
Prescription
First Approved
1988-12-20
Routes
ORAL
Dosage Forms
TABLET

Companies

Active Ingredient: CLOMIPHENE CITRATE

MILOPHENE Approval History

1989
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2026
Original
New Indication
New Form
Label Update
7 FDA actions from 1988 to 2025
Aug 2025 SUPPL
Mfg · Manufacturing (CMC)
Jan 1998 SUPPL
Mfg · Manufacturing (CMC)
Dec 1988 ORIGINAL
Update

What MILOPHENE Treats

5 indications

MILOPHENE is approved for 5 conditions since its original approval in 1988. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Ovulatory Dysfunction
  • Polycystic Ovary Syndrome
  • Amenorrhea-Galactorrhea Syndrome
  • Psychogenic Amenorrhea
  • Secondary Amenorrhea
Source: FDA Label

MILOPHENE Competitive Set

Pro

Three rings of competition based on shared molecular targets and treated indications.

Indication competitors

2

Same indication, different mechanism — what else might this patient receive?

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to MILOPHENE

3 of 4

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

CLOMIPHENE CITRATE
CLOMIPHENE CITRATE
5 shared
ACCORD HLTHCARE
Shared indications:
Ovulatory DysfunctionPolycystic Ovary SyndromeAmenorrhea-Galactorrhea Syndrome +2 more
CRINONE
PROGESTERONE
1 shared
WATSON LABS INC
Shared indications:
Secondary Amenorrhea
NORETHINDRONE ACETATE
NORETHINDRONE ACETATE
1 shared
Teva
Shared indications:
Secondary Amenorrhea
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Clinical Trial Registry

32 trials
Trial Sponsor ID Phase Status Title
NCT03059173 MYOPK 2015_68 2016-A01246-45, PHRC_N_15-0116 Ph 3 recruiting Interest of Myo-inositol Supplementation in Women With Polycystic Ovarian Syndrome
NCT04944836 RCRHRT Ph 2 recruiting Sex Hormone Supplementation and Rotator Cuff Repair: A Preliminary Randomized Trial
NCT06701071 HS-23-00039 Ph 4 recruiting Evaluation of a Long Versus Short Clomid Protocol for Controlled Ovarian Stimulation
NCT05206448 CLC II results posted 201906826 Ph 4 active not recruiting Randomized Controlled Trial of Combined Letrozole and Clomid (CLC II) Versus Letrozole Alone for Women With Anovulation
NCT06564961 4068 Ph 3 completed Clomiphene Citrate in Infertile Men With Idiopathic Oligoasthenozoospermia
NCT00427700 results posted RACLO Ph 3 completed Induction of Ovulation With Raloxifene or Clomiphene Citrate in Polycystic Ovarian Syndrome
NCT02523898 SemnanUMS1 Ph 2 terminated Metformine and CC Compared With Placebo and CC for Induction Ovulation in PCOS Patients With Insulin Resistant
NCT02436226 MT1 Ph 4 completed Use of Low Dose of HCG During Ovulation Induction With CC in Women With CC Resistant PCOS
NCT05231980 86 Ph 2 completed Efficacy of Pentoxifylline and Alpha Lipoic Acid in PCOS Resistant to Clomiphene Citrate
NCT04177693 results posted 2000028370 1R01HD100369-01 Ph 1 completed Pharmacokinetics and Hepatic Safety of EGCG
NCT04306692 2018-004604-20 Ph 4 terminated Myo-inositol Versus Clomiphene Citrate in PCOS
NCT04210765 2019.08.1.04.061 Ph 4 completed Incremental Clomiphene Citrate Doses in Successive Cycles and FSH, LH and Steroid Hormone Levels
NCT04302532 1 Ph 4 completed Coenzyme q 10 and Fertility Outcome in Women With Clomiphene Resistant PCOS
NCT03674385 PHCL 191 Ph 2 completed Efficacy of Vit E in PCOS Resistant to Clomiphene Citrate
NCT03770026 181210 Ph 2, Ph 3 completed Autologous Platelet-rich Plasma for Clomiphene Citrate-induced Thin Endometrium
NCT02274311 results posted ClomipheneAcro Ph 2 completed Clomiphene Citrate for Treatment of Acromegaly
NCT01880086 results posted Cornell-1301013472 Ph 2 completed Clomiphene Citrate for the Treatment of Low Testosterone Associated With Chronic Opioid Pain Medication Administration
NCT00719186 PPCOSII results posted RMN-PPCOSII Ph 3 completed Pregnancy in Polycystic Ovary Syndrome II
NCT01008319 Clomid results posted 2078 Ph 3 completed Traditional Clomiphene Citrate Administration vs. Stair-step Approach
NCT02380755 385.615 2013/16781-1 Ph 2 completed Clomiphene Citrate for the Treatment of Obesity Related Male Hypogonadism
NCT02775734 NAC AS1275 Ph 2, Ph 3 completed NAC in CC Resistant PCOS After LOD
NCT02352597 PCOS 222 Ph 4 completed Phytoestrogens as an Alternative to Estradiol in Ovulation Induction in PCOS
NCT02381184 khalid-walid Ph 2, Ph 3 completed Extended Clomiphene Citrate Regimen in Women With Polycystic Ovary Syndrome
NCT02479256 20092009 Ph 4 completed Clomiphene Citrate Versus Tamoxifen for Ovulation Induction in PCOs
NCT00796289 2008-03 Ph 2 completed Study to Assess the Efficacy and Safety of Three Dosage Strengths of Pulsatile GnRH Delivered From a Iontophoretic Patch Compared to Oral Treatment With Clomiphene or Placebo in Infertile Females
NCT01638988 OVO-12-17 Ph 3 withdrawn Clomifene Citrate Versus Metformin in First-line Treatment of Infertility in Patients With Polycystic Ovary Syndrome and a Resistance to Insulin
NCT01044862 AMIGOS results posted RMN-AMIGOS 3U10HD055925-02S1, 5U10HD055925 Ph 3 completed Assessment of Multiple Intrauterine Gestations From Ovarian Stimulation
NCT00501839 05/2006a Ph 4 withdrawn Clomiphene Citrate in Infertile PCOS Patients
NCT00835744 cc versus FSH 2008/192 Ph 4 completed Comparison of Clomiphene Citrate and Gonadotropins in Ovulation Induction Cycles
NCT01004068 06/2009 Ph 4 completed Short-term Structured Exercise Training Program Plus Diet Intervention in Patients With Polycystic Ovary Syndrome (PCOS)
NCT01213147 2063 Ph 4 completed Mild Stimulation Protocol Versus Microdose Gonadotropin-releasing Hormone Agonist Flare up Protocol in Poor Responders
NCT00830492 YazdRCCI1388 Ph 4 completed Clomiphene Citrate (CC)/Gonadotropin/Gonadotropin Releasing Hormone (GnRH) Antagonist Versus Gonadotropin/GnRH Agonist
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Active Pipeline

Pro

Ongoing clinical trials by development phase

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Key Completed Trials

Pro

Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

MILOPHENE FDA Label Details

Indications & Usage

MILOPHENE is indicated for the treatment of Ovulatory Dysfunction; Polycystic Ovary Syndrome; Amenorrhea-Galactorrhea Syndrome; Psychogenic Amenorrhea; Secondary Amenorrhea.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment