TheraRadar
Data updated: May 26, 2026

TROGARZO (ibalizumab-uiyk)

CD4-directed Antibody Interactions Trial Activity: Declining
First-in-Class Orphan Drug Breakthrough Therapy Priority Review Fast Track
Infectious Disease Approved 2018-03-06

TROGARZO is indicated for the treatment of Human Immunodeficiency Virus Infection.

Source: FDA Label • THERATECHNOLOGIES • CD4-directed Blocking Antibody

How TROGARZO Works

Trogarzo is a CD4-directed blocking antibody that functions as a post-attachment HIV-1 inhibitor. It targets the CD4 receptor on host cells to interfere with the viral infection process. By acting as a fusion inhibitor after the virus has already bound to the cell, the medication prevents HIV-1 from successfully entering and infecting the host cell.

Development Insights

TaiMed Biologics Inc. conducting 5 trials (100%)
2 indications explored (Focused)
hiv (4 trials)
hiv-1-infection (1 trials)
2
Indications
--
Phase 3 Trials
1
Priority Reviews
8
Years on Market

Details

Status
Prescription
First Approved
2018-03-06
Patent Cliff
2025

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Routes
INJECTION
Dosage Forms
INJECTABLE

Companies

Active Ingredient: IBALIZUMAB-UIYK

TROGARZO Approval History

2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
6 FDA actions from 2018 to 2023 · 1 indication expansions
Dec 2023 SUPPL
Label · Labeling
Oct 2022 SUPPL
Efficacy
Apr 2021 SUPPL
Label · Labeling

What TROGARZO Treats

1 indications

TROGARZO is approved for 1 conditions since its original approval in 2018. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Human Immunodeficiency Virus Infection
Source: FDA Label

TROGARZO Competitive Set

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Three rings of competition based on shared molecular targets and treated indications.

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to TROGARZO

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Clinical Trial Registry

4 trials
Trial Sponsor ID Phase Status Title
NCT03913195 results posted TMB-302 Ph 3 completed Study of the Safety of Trogarzo™ Administered as an Undiluted "IV Push" or an Intramuscular Injection
NCT02707861 results posted TMB-311 Ph 3 completed Ibalizumab Plus Optimized Background Regimen in Treatment-Experienced Patients With Multi-Drug Resistant HIV-1
NCT02475629 results posted TMB-301 Ph 3 completed Ibalizumab Plus Optimized Background Regimen in Patient With Multi-Drug Resistant HIV
NCT00784147 TMB-202 results posted TMB-202 Amendment 2 Ph 2 completed Dose-Response Study of Ibalizumab (Monoclonal Antibody) Plus Optimized Background Regimen in Patients With HIV-1
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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

TROGARZO FDA Label Details

Indications & Usage

FDA Label (PDF)

TROGARZO is indicated for the treatment of Human Immunodeficiency Virus Infection.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment