TheraRadar
Data updated: May 26, 2026

ZINPLAVA (bezlotoxumab)

Trial Activity: Mature
First-in-Class
Infectious Disease Approved 2016-10-21

ZINPLAVA is indicated for the treatment of Clostridioides Difficile Infection.

Source: FDA Label • Merck

How ZINPLAVA Works

ZINPLAVA is a human monoclonal antibody that targets and binds to Clostridioides difficile toxin B. By binding to this specific toxin, the drug neutralizes its harmful biological effects. This action helps to prevent the recurrence of the infection in patients already undergoing antibacterial treatment. It does not directly target the bacteria itself, but rather the toxins produced by the pathogen.

Development Insights

Hellenic Institute for the Study of Sepsis conducting 1 trials (13%)
17 indications explored (Broad Platform)
inflammatory bowel diseases (2 trials)
clostridium difficile infection (2 trials)
clostridioides difficile infection (1 trials)
2
Indications
--
Phase 3 Trials
2
Priority Reviews
9
Years on Market

Details

Status
Prescription
First Approved
2016-10-21
Routes
INJECTION
Dosage Forms
INJECTABLE

Companies

Active Ingredient: BEZLOTOXUMAB

ZINPLAVA Approval History

2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
2 FDA actions from 2016 to 2023 · 1 indication expansions
May 2023 SUPPL Priority
Efficacy
Oct 2016 ORIGINAL Priority
New Drug · Type 1 - New Molecular Entity

What ZINPLAVA Treats

1 indications

ZINPLAVA is approved for 1 conditions since its original approval in 2016. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Clostridioides Difficile Infection
Source: FDA Label

ZINPLAVA Competitive Set

Pro

Three rings of competition based on shared molecular targets and treated indications.

Indication competitors

2

Same indication, different mechanism — what else might this patient receive?

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

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Clinical Trial Registry

8 trials
Trial Sponsor ID Phase Status Title
NCT05304715 BEYOND results posted BEYOND 2021-005473-10 Ph 2 completed Bezlotoxumab Yielded Outcomes by Addressing Personalized Needs in Clostridioides Difficile Infection
NCT03829475 ICON-2 results posted 2018 Ph 2 completed ICON-2: FMT and Bezlotoxumab Compared to FMT and Placebo for Patients With IBD and CDI
NCT04626947 results posted STUDY19100301 Ph 4 terminated Prevention of Recurrent Clostridium Difficile Infection (CDI) in Patients With Inflammatory Bowel Disease (IBD).
NCT03182907 MODIFY III results posted 6072-001 MK-6072-001, 2017-000070-11 Ph 3 completed Bezlotoxumab (MK-6072) Versus Placebo in Children With Clostridium Difficile Infection (CDI) (MK-6072-001)
NCT03756454 2018H0348 Ph 4 terminated Comparing the Effectiveness of IV Bezlotoxumab Versus Placebo in Decreasing Morbidity and Mortality in Patients With Fulminant C. Diff Requiring Surgery.
NCT05077085 BSTEP BSTEP Ph 4 withdrawn Bezlotoxumab Versus FMT for Multiple Recurrent CDI
NCT03937999 results posted 2019-10212 Ph 4 terminated Bezlotoxumab as Secondary Prophylaxis for C. Difficile in High-risk Hospitalized Patients Exposed to Antibiotics.
NCT03880539 BEZLO Study00143405 Ph 4 completed Bezlotoxumab (BEZLO) In Addition To Standard Of Care (SOC) Vancomycin For The Treatment of Multi-Recurrent Clostridium Difficile Infection
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Active Pipeline

Pro

Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

ZINPLAVA FDA Label Details

Indications & Usage

FDA Label (PDF)

ZINPLAVA is indicated for the treatment of Clostridioides Difficile Infection.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment