TheraRadar
Data updated: May 26, 2026

ZULRESSO (brexanolone)

Trial Activity: Stable 2 active trials
First-in-Class Breakthrough Therapy Priority Review
CNS Approved 2019-03-19

Development Insights

Supernus Pharmaceuticals, Inc. conducting 3 trials (38%)
10 indications explored (Broad Platform)
postpartum depression (2 trials)
depression (1 trials)
ptsd (1 trials)
2
Indications
--
Phase 3 Trials
2
Priority Reviews
7
Years on Market

Details

Status
Discontinued
First Approved
2019-03-19
Patent Cliff
2037

Pro Metrics

Patent cliff and revenue data

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Routes
INTRAVENOUS
Dosage Forms
SOLUTION

Companies

Active Ingredient: BREXANOLONE

ZULRESSO Approval History

2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
9 FDA actions from 2019 to 2025 · 1 indication expansions
Jan 2025 SUPPL
Update · REMS
Oct 2023 SUPPL
Update · REMS
Mar 2023 SUPPL
Update · REMS

What ZULRESSO Treats

2 FDA approvals

Originally approved for its first indication in 2019 . Covers 2 distinct patient populations.

  • Other (2)
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Clinical Trial Registry

7 trials
Trial Sponsor ID Phase Status Title
NCT05329779 results posted 2021P003137 Ph 4 terminated Study on Allopregnanolone and Depression in Perimenopausal Women
NCT05223829 2000031354 U54AA027989 Ph 1 active not recruiting Utility of Brexanolone to Target Stress-induced Alcohol Use Among Men and Women With Posttraumatic Stress Disorder
NCT05645432 results posted 547-TRM-201 Ph 2 completed An Open-Label Study Evaluating Brexanolone in Adults With Tinnitus
NCT03665038 results posted 547-PPD-304 2017-004356-34 Ph 3 completed A Study to Assess the Safety of Brexanolone in the Treatment of Adolescent Female Participants With Postpartum Depression (PPD)
NCT06580444 AS210006-A09 Ph 2 not yet recruiting Brexanolone to Target Concurrent PTSD and Stress Induced Alcohol Use in Veterans: A Dose Finding Study
NCT04537806 results posted 547-ARD-301 Ph 3 terminated A Study of Brexanolone for Acute Respiratory Distress Syndrome (ARDS) Due to Coronavirus Disease 2019 (COVID-19)
NCT04273191 547-EXM-401 Ph 4 withdrawn A Study to Evaluate Multimodal Neuroimaging Parameters in Women With Postpartum Depression Who Are Receiving ZULRESSO™ (Brexanolone)
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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

ZULRESSO FDA Label Details

View full patent landscape →
8 OB patents · 4 families · 205 international docs across 32 countries

ZULRESSO Patents & Exclusivity

Latest Patent: Mar 2037

Patents (8 active)

US10940156 Expires Mar 8, 2037
US10251894 Expires Nov 27, 2033
US10322139 Expires Jan 23, 2033
US8410077 Expires Mar 13, 2029
US9200088 Expires Mar 13, 2029
US9750822 Expires Mar 13, 2029
US7635773 Expires Mar 13, 2029
US10117951 Expires Mar 13, 2029
Source: FDA Orange Book

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Deep insights for ZULRESSO

Revenue Insights

  • Quarterly revenue tracking
  • Historical trend analysis

Patent Timeline

  • Cliff: 2037
  • 8 active patents

Trial Analysis

  • 8 total trials
  • Stage: Stable

Competitive Landscape

  • Competitor tracking
  • Same target/indication analysis
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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment