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Data updated: May 26, 2026

ATOVAQUONE AND PROGUANIL HYDROCHLORIDE (atovaquone)

Infectious Disease Approved 2011-01-12

Atovaquone and proguanil hydrochloride is an antimalarial medication used to prevent Plasmodium falciparum malaria, even in geographic regions where chloroquine resistance is common. It also treats patients with acute, uncomplicated cases of the infection. This combination is particularly useful in areas where other standard treatments, such as mefloquine or halofantrine, may fail due to drug resistance.

Source: FDA Label • GLENMARK PHARMS LTD • Antimalarial

How ATOVAQUONE AND PROGUANIL HYDROCHLORIDE Works

This medication works by combining atovaquone and proguanil hydrochloride into a single fixed-dose tablet. Together, these components function as an antiprotozoal agent to target and eliminate the Plasmodium falciparum parasite.

Source: FDA Label
2
Indications
--
Phase 3 Trials
15
Years on Market

Details

Status
Prescription
First Approved
2011-01-12
Routes
ORAL
Dosage Forms
TABLET

ATOVAQUONE AND PROGUANIL HYDROCHLORIDE Approval History

2012
2013
2014
2015
2016
2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
10 FDA actions from 2011 to 2019
Nov 2019 SUPPL
Label · Labeling
Jun 2014 SUPPL
Label · Labeling
May 2014 ORIGINAL
Update

What ATOVAQUONE AND PROGUANIL HYDROCHLORIDE Treats

1 indications

ATOVAQUONE AND PROGUANIL HYDROCHLORIDE is approved for 1 conditions since its original approval in 2011. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Malaria
Source: FDA Label

ATOVAQUONE AND PROGUANIL HYDROCHLORIDE Competitive Set

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📋

Clinical Trial Registry

4 trials
Trial Sponsor ID Phase Status Title
NCT07357103 SPIRIT-ALT 2026-12268 527077 Ph 4 not yet recruiting Positioning Second-line Therapies for Pneumocystis Jirovecii Pneumonia (PCP Alternatives)
NCT05998135 STUDY00005363 NCI-2023-03479, STUDY00005363 Ph 2 recruiting Repurposing Atovaquone for the Treatment of Platinum-Resistant Ovarian Cancer
NCT06624371 AflacBT2303 STUDY00007693 Ph 1 recruiting Atovaquone Combined With Radiation in Children With Malignant Brain Tumors
NCT01858831 116441 Ph 1 completed Single Oral Dose Study of Atovaquone/Proguanil Hydrochloride Combination Tablets and Atovaquone Suspension
🔬

Active Pipeline

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Key Completed Trials

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Completed studies with published results, ranked by significance

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📊

Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

ATOVAQUONE AND PROGUANIL HYDROCHLORIDE FDA Label Details

Indications & Usage

ATOVAQUONE AND PROGUANIL HYDROCHLORIDE is indicated for the treatment of Malaria.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.