TheraRadar
Data updated: May 26, 2026

HUMULIN R KWIKPEN (insulin human)

Trial Activity: Stable 2 active trials
Metabolic Approved 1982-10-28

AFREZZA is a rapid-acting inhaled human insulin indicated to improve glycemic control in adult patients with diabetes mellitus. As an inhaled formulation, it provides a method for managing blood sugar levels without the need for traditional injection. The medication is not recommended for the treatment of diabetic ketoacidosis or for use in patients who currently smoke or have recently stopped smoking.

Source: FDA Label • Eli Lilly • Insulin

How HUMULIN R KWIKPEN Works

This medication lowers blood glucose levels by stimulating peripheral glucose uptake in skeletal muscle and fat tissues. It further regulates blood sugar by inhibiting the liver's production of glucose. Additionally, the drug inhibits the breakdown of fats and proteins while simultaneously enhancing protein synthesis within the body.

Development Insights

Columbia University conducting 3 trials (43%)
12 indications explored (Broad Platform)
insulin resistance (3 trials)
non-alcoholic fatty liver disease (3 trials)
prediabetic state (3 trials)
3
Indications
--
Phase 3 Trials
43
Years on Market

Details

Status
Prescription
First Approved
1982-10-28
Routes
SUBCUTANEOUS
Dosage Forms
SOLUTION

Companies

Active Ingredient: INSULIN HUMAN

HUMULIN R KWIKPEN Approval History

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Original
New Indication
New Form
Label Update
102 FDA actions from 1982 to 2022 · 2 indication expansions
Jun 2022 SUPPL
Label · Labeling
Nov 2019 SUPPL
Label · Labeling
Aug 2019 SUPPL
Label · Labeling

What HUMULIN R KWIKPEN Treats

1 indications

HUMULIN R KWIKPEN is approved for 1 conditions since its original approval in 1982. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Diabetes
Source: FDA Label

HUMULIN R KWIKPEN Boxed Warning

RISK OF ACUTE BRONCHOSPASM IN PATIENTS WITH CHRONIC LUNG DISEASE Acute bronchospasm has been observed in AFREZZA-treated patients with asthma and Chronic Obstructive Pulmonary Disease (COPD) [see Warnings and Precautions ( 5.1 )]. AFREZZA is contraindicated in patients with chronic lung disease such as asthma or COPD [see Contraindications ( 4 )]. Before initiating AFREZZA, perform a detailed medical history, physical examination, and spirometry (FEV 1 ) to identify potential lung disease in all...

HUMULIN R KWIKPEN Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

What's emerging in HUMULIN R KWIKPEN's indications

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Phase 3 candidates targeting molecules with no FDA-approved drug, in indications HUMULIN R KWIKPEN treats. First-in-class if their pivotal trials read out positive.

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Clinical Trial Registry

6 trials
Trial Sponsor ID Phase Status Title
NCT06558422 AAAU9702 P30DK063608, K12DK133995 Ph 1 not yet recruiting Human Models of Selective Insulin Resistance: Pancreatic Clamp
NCT05724134 AAAU3014 3P30DK063608 Ph 1 completed Pancreatic Clamp in NAFLD
NCT06939959 579/DME/KMC Ph 4 recruiting Evaluating the Efficacy of Topical Insulin for the Restoration of Ocular Surface Interface in Dry Eye Disease.
NCT06126354 AAAU7680 3P30DK063608 Ph 1 withdrawn Dexamethasone/Pancreatic Clamp P&F
NCT02028078 PILOT_EGP PILOT_EGP Ph 2 completed Pilot Study Investigating the Feasibility of Determining the Endogenous Glucose Production During a Hypoglycaemia
NCT01269606 ANA-3877 U1111-1117-1353, JapicCTI-111383 Ph 1 completed Comparing Insulin Aspart With Fast-acting Insulin Human in Subjects With Type 1 Diabetes
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Active Pipeline

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

HUMULIN R KWIKPEN FDA Label Details

Indications & Usage

FDA Label (PDF)

HUMULIN R KWIKPEN is indicated for the treatment of Diabetes.

⚠️ BOXED WARNING

WARNING: RISK OF ACUTE BRONCHOSPASM IN PATIENTS WITH CHRONIC LUNG DISEASE Acute bronchospasm has been observed in AFREZZA-treated patients with asthma and Chronic Obstructive Pulmonary Disease (COPD) [see Warnings and Precautions ( 5.1 )]. AFREZZA is contraindicated in patients with chronic lung dis...

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment