TheraRadar
Data updated: May 26, 2026

INBRIJA (levodopa)

CNS Approved 2018-12-21

INBRIJA is an aromatic amino acid indicated for the intermittent treatment of OFF episodes in patients with Parkinson's disease. This medication is specifically for patients who are already receiving treatment with carbidopa/levodopa. It serves as a supplemental therapy to address the return of symptoms that occurs between scheduled doses of maintenance medication.

Source: FDA Label • MERZ • Aromatic Amino Acid

How INBRIJA Works

Levodopa functions as a metabolic precursor to dopamine, a chemical messenger in the brain. The drug crosses the blood-brain barrier and is presumably converted into dopamine within the central nervous system. This process is thought to be the mechanism by which the medication relieves the symptoms associated with Parkinson's disease.

1
Indication
--
Phase 3 Trials
7
Years on Market

Details

Status
Prescription
First Approved
2018-12-21
Patent Cliff
2033

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Routes
INHALATION
Dosage Forms
POWDER

Companies

Active Ingredient: LEVODOPA

INBRIJA Approval History

2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
5 FDA actions from 2018 to 2026
Mar 2026 SUPPL
Label · Labeling
Aug 2020 SUPPL
Label · Labeling
Aug 2019 SUPPL
Label · Labeling

What INBRIJA Treats

1 indications

INBRIJA is approved for 1 conditions since its original approval in 2018. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Parkinson's Disease
Source: FDA Label

INBRIJA Competitive Set

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Three rings of competition based on shared molecular targets and treated indications.

Indication competitors

2

Same indication, different mechanism — what else might this patient receive?

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

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Clinical Trial Registry

17 trials
Trial Sponsor ID Phase Status Title
NCT02601586 OXYDOPA 14 7440 01 Ph 2, Ph 3 completed Effects of PR Oxycodone and of Levodopa, vs Placebo, on Central Neuropathic Pain in Parkinson's Disease
NCT06234995 STUDY00007291 P50NS123103, 2025P008808 Ph 4 recruiting Cortical Electrophysiology of Response Inhibition in Parkinson's Disease
NCT07444892 STUDY00002995 2025P013031 Ph 2 completed Levodopa for Diabetic Retinopathy
NCT03000569 results posted 217-PRK-201 Ph 2 completed A Study to Evaluate SAGE-217 in Participants With Parkinson's Disease
NCT02744391 results posted 7270 Ph 4 completed A Study of L-DOPA for Depression and Slowing in Older Adults
NCT03205956 MPDP 009 Ph 1 completed Measuring Parkinson's Disease Progression
NCT03055936 COMDOS1 results posted 3112005 Ph 1 completed Dose-finding Pharmacokinetic Study in Healthy Males
NCT02769793 16-2015-52 Ph 4 completed Efficacy of Levodopa/Benserazide Dispersible Tablet on Response Fluctuations in PD Patients With Delayed ON
NCT01281475 results posted 09-12-0610 3523 Ph 2, Ph 3 completed A Trial of Levodopa in Angelman Syndrome
NCT02560389 results posted 204583 Ph 4 completed Dopamine Enhancement of Fear Extinction Learning in PTSD (1R21MH108753)
NCT00845000 results posted P05550 MK-3814-023 Ph 1 completed Acute Effects of Preladenant (SCH 420814) on Dyskinesia and Parkinsonism in Levodopa Treated Participants (P05550)
NCT01176435 results posted 0912M75653 Ph 2 completed Trial of L-DOPA as a Treatment to Improve Vision in Albinism
NCT00713583 results posted 1R01DA023608-01 1R01DA023608-01, R01DA023608-01 Ph 2 completed Carbidopa/Levodopa Combined With Behavioral Therapy for the Treatment of Cocaine Dependence
NCT02641054 CT-CVXL-0107-01 Ph 2 completed Efficacy Phase IIa Study of CVXL-0107 in Advanced Parkinson's Disease
NCT02073773 CIRB 2013/323/D Ph 3 completed Combinational Rehabilitative Therapy and Functional Brain Imaging for Patients Recovering From Motor Stroke
NCT01227655 BIPARKII results posted BIA-91067-302 2010-022366-27, BIA-91067-302 Ph 3 completed Efficacy and Safety of BIA 9-1067 in Idiopathic Parkinson's Disease Patients.
NCT01568073 results posted BIA-91067-301 2010-021860-13 Ph 3 completed Efficacy and Safety of BIA 9-1067 in Idiopathic Parkinson's Disease Patients With "Wearing-off" Phenomenon
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Active Pipeline

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Key Completed Trials

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Trial Timeline

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

INBRIJA FDA Label Details

Indications & Usage

FDA Label (PDF)

INBRIJA is indicated for the treatment of Parkinson's Disease.

View full patent landscape →
6 OB patents · 3 families · 84 international docs across 22 countries

INBRIJA Patents & Exclusivity

Latest Patent: Oct 2033

Patents (6 active)

US12458615 Expires Oct 21, 2033
US8685442 Expires Nov 16, 2032
US8945612 Expires Nov 16, 2032
US8545878 Expires Nov 16, 2032
US9393210 Expires Nov 16, 2032
USRE43711 Expires Feb 3, 2029
Source: FDA Orange Book

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Revenue Insights

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Patent Timeline

  • Cliff: 2033
  • 6 active patents

Trial Analysis

  • Clinical trial tracking
  • Development stage analysis

Competitive Landscape

  • 20 similar drugs
  • Same target/indication analysis
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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.