TheraRadar
Data updated: May 26, 2026

IWILFIN (eflornithine hydrochloride)

Oncology Approved 2023-12-13

Iwilfin is indicated to reduce the risk of relapse in adult and pediatric patients with high-risk neuroblastoma (HRNB). It is used as maintenance therapy for patients who have demonstrated at least a partial response to prior multiagent, multimodality therapy, including anti-GD2 immunotherapy. By addressing minimal residual disease, the drug helps prevent or delay the return of the cancer following intensive primary treatment.

How IWILFIN Works

Eflornithine is an irreversible inhibitor of ornithine decarboxylase (ODC), the rate-limiting enzyme in polyamine biosynthesis and a transcriptional target of MYCN. Polyamines are essential for neoplastic transformation and cell proliferation. By inhibiting polyamine synthesis, eflornithine decreases the expression of oncogenic drivers MYCN and LIN28B and restores the balance of the LIN28/Let-7 metabolic pathway, which regulates cancer stem cells. This results in a cytostatic effect that suppresses neurosphere formation and delays tumor recurrence.

1
Indication
--
Phase 3 Trials
1
Priority Reviews
2
Years on Market

Details

Status
Prescription
First Approved
2023-12-13
Patent Cliff
2036

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Routes
ORAL
Dosage Forms
TABLET

Companies

Active Ingredient: EFLORNITHINE HYDROCHLORIDE

IWILFIN Approval History

2024
2025
2026
Original
New Indication
New Form
Label Update
2 FDA actions from 2023 to 2024
Nov 2024 SUPPL
Label · Labeling
Dec 2023 ORIGINAL Priority
Update · Type 5 - New Formulation or New Manufacturer

What IWILFIN Treats

1 indications

IWILFIN is approved for 1 conditions since its original approval in 2023. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Neuroblastoma
Source: FDA Label

IWILFIN Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to IWILFIN

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FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

ADREVIEW
IOBENGUANE SULFATE I-123
1 shared
GE HEALTHCARE
Shared indications:
Neuroblastoma
CYCLOPHOSPHAMIDE
CYCLOPHOSPHAMIDE
1 shared
Hikma
Shared indications:
Neuroblastoma
CYTOXAN
CYCLOPHOSPHAMIDE
1 shared
Baxter
Shared indications:
Neuroblastoma
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Clinical Trial Registry

1 trials
Trial Sponsor ID Phase Status Title
NCT03794349 results posted ANBL1821 NCI-2018-03377, ANBL1821 Ph 2 active not recruiting Irinotecan Hydrochloride, Temozolomide, and Dinutuximab With or Without Eflornithine in Treating Patients With Relapsed or Refractory Neuroblastoma
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Active Pipeline

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

IWILFIN FDA Label Details

Indications & Usage

FDA Label (PDF)

IWILFIN is indicated for the treatment of Neuroblastoma.

IWILFIN Patents & Exclusivity

Latest Patent: Feb 2036
Exclusivity: Dec 2030

Patents (1 active)

US12582625 Expires Feb 12, 2036

Exclusivity

NP Until Dec 2026
ODE-462 Until Dec 2030
Source: FDA Orange Book

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Revenue Insights

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Patent Timeline

  • Cliff: 2036
  • 1 active patents

Trial Analysis

  • Clinical trial tracking
  • Development stage analysis

Competitive Landscape

  • 9 similar drugs
  • Same target/indication analysis
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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.