TheraRadar
Data updated: May 26, 2026

LOPID (gemfibrozil)

Peroxisome Proliferator-activated Receptor alpha Agonists Trial Activity: Declining 1 active trials
Cardiovascular Approved 1981-12-21

LOPID is indicated for the treatment of Hypertriglyceridemia; Pancreatitis.

Source: FDA Label • Pfizer

Development Insights

Bristol-Myers Squibb conducting 2 trials (10%)
17 indications explored (Broad Platform)
healthy participants (3 trials)
healthy (3 trials)
healthy subjects (3 trials)
2
Indications
--
Phase 3 Trials
44
Years on Market

Details

Status
Prescription
First Approved
1981-12-21
Routes
ORAL
Dosage Forms
TABLET, CAPSULE

Companies

Active Ingredient: GEMFIBROZIL

LOPID Approval History

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Original
New Indication
New Form
Label Update
132 FDA actions from 1981 to 2020 · 1 indication expansions
Dec 2020 SUPPL
Label · Labeling
Apr 2018 SUPPL
Label · Labeling
Apr 2017 SUPPL
Label · Labeling

What LOPID Treats

2 indications

LOPID is approved for 2 conditions since its original approval in 1981. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Hypertriglyceridemia
  • Pancreatitis
Source: FDA Label

LOPID Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

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CHOLESTYRAMINE
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Shared indications:
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Clinical Trial Registry

21 trials
Trial Sponsor ID Phase Status Title
NCT05931484 FHL-301-001 Ph 2 not yet recruiting Study to Evaluate the Safety, Tolerability, Efficacy, and PK of FHL-301 in Parkinson's Disease Patients.
NCT06064539 INT16726 U1111-1244-2759 Ph 1 completed Study of Drug-drug Interaction of the Effects of Gemfibrozil and Rifampicin on SAR442168 in Healthy Adult Subjects
NCT06809608 BP45670 2024-517360-37-00 Ph 1 completed A Study Investigating the Effect of Different Approved Medications on How the Body Processes the Study Compound RO7795081
NCT05959447 results posted 221854 BUS-P1-12 Ph 1 completed Evaluation of the Potential Drug-drug Interactions Between Gemfibrozil or Dabigatran Etexilate and Camlipixant
NCT02770222 AC-065-113 2016-000811-34 Ph 1 completed A Clinical Study to Investigate the Effect of Gemfibrozil or Rifampicin on Blood Concentrations of Selexipag in Healthy Subjects
NCT06392659 VX24-993-004 Ph 1 completed A Phase 1, Open-label Study Evaluating the Pharmacokinetics and Drug-drug Interaction of VX-993 in Healthy Adults
NCT05932303 IM027-1007 Ph 1 completed A Study to Assess the Effect of Multiple Doses of Itraconazole, Gemfibrozil, or Carbamazepine on BMS-986278 in Healthy Participants
NCT04956627 IM018-004 Ph 1 completed A Study to Assess the Effect of Itraconazole, Phenytoin and Gemfibrozil on the Drug Levels of BMS-986166 in Healthy Participants
NCT03723395 ONT-380-012 Ph 1 completed A Drug-Drug Interaction Study in Healthy Volunteers of the Effects of Tucatinib
NCT03624959 RPC01-1912 U1111-1215-6965 Ph 1 completed Drug-drug Interaction Study of Ozanimod With Inhibitor or Inducer of CYP2C8 and/or CYP3A
NCT01836198 results posted 14586 I1R-MC-GLBZ Ph 1 completed The Effect of Gemfibrozil, Ketoconazole and Clarithromycin on the Amount of LY2409021 in the Bloodstream
NCT02638597 GEMNIC results posted STU 072014-088 Ph 2 completed Gemfibrozil for Nicotine Smoking Cessation
NCT01736254 results posted 14701 I1V-MC-EIBD Ph 1 completed A Study of Evacetrapib in Healthy Participants
NCT01340846 113771 Ph 1 completed A Pharmacokinetics Study of the Effects of GSK2118436 on Warfarin, the Effects of Ketoconazole and Gemfibrozil on GSK2118436, and the Effects of Repeat Doses of GSK2118436 in Subjects With BRAF Mutant Solid Tumors
NCT01376232 DDI 113634 Ph 1 completed Study to Assess the Pharmacokinetics of GSK1278863A Coadministered With a High Fat Meal or an Inhibitor of CYP2C8 (Gemfibrozil)
NCT01876810 results posted 082/2012 Ph 2 completed Initial Screening of Gemfibrozil as a Novel Treatment for Tobacco Addiction
NCT02230033 CR105398 56021927PCR1012 Ph 1 completed Study to Assess Drug-Drug Interaction Between Itraconazole or Gemfibrozil and JNJ-56021927
NCT01301742 results posted 1245.58 2010-023152-85 Ph 1 completed Relative Bioavailability of Single Dose Empagliflozin (BI 10773) When Co-administered With Multiple Doses of 600 mg Gemfibrozil Compared to Single Dose Treatment With Empagliflozin (BI 10773) When Given Alone in Healthy Volunteers
NCT01913379 9785-CL-0006 2011-000333-37 Ph 1 completed Drug-drug Interaction Study With MDV3100 (ASP9785) and Gemfibrozil and Itraconazole
NCT01797198 3652-CL-0006 2011-002874-21 Ph 1 completed A Study to Assess the Effect of Multiple Doses of Gemfribozil on a Single Dose of ASP3652, and to Assess the Effects of Multiple Doses of ASP3652 on a Single Dose of Repaglinide in the Body of Healthy Subjects
NCT01083212 D1020C00030 Ph 1 completed To Evaluate the Effect of Gemfibrozil on the Pharmacokinetics and Pharmacodynamics of a Single Dose of AZD1656
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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

LOPID FDA Label Details

Indications & Usage

FDA Label (PDF)

LOPID is indicated for the treatment of Hypertriglyceridemia; Pancreatitis.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment