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Data updated: May 26, 2026

METHYLIN ER (methylphenidate hydrochloride)

CNS Approved 2000-05-09

Methylin ER is an extended-release medication used for children aged 6 to 12 who have Attention Deficit Hyperactivity Disorder (ADHD). As a central nervous system stimulant, it helps patients in this age group manage their symptoms. It is prescribed to provide long-acting support for pediatric patients dealing with the challenges of ADHD.

Source: FDA Label • SPECGX LLC

How METHYLIN ER Works

This medication works by stimulating the central nervous system. While it is classified as a stimulant, the specific process by which it produces a therapeutic effect for ADHD is not currently known.

Source: FDA Label
1
Indication
--
Phase 3 Trials
26
Years on Market

Details

Status
Prescription
First Approved
2000-05-09
Routes
ORAL
Dosage Forms
TABLET, EXTENDED RELEASE

Companies

Active Ingredient: METHYLPHENIDATE HYDROCHLORIDE

METHYLIN ER Approval History

2001
2002
2003
2004
2005
2006
2007
2008
2009
2010
2011
2012
2013
2014
2015
2016
2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
26 FDA actions from 2000 to 2025
Oct 2025 SUPPL
Label · Labeling
Oct 2025 SUPPL
Label · Labeling
Jun 2021 SUPPL
Label · Labeling

What METHYLIN ER Treats

1 indications

METHYLIN ER is approved for 1 conditions since its original approval in 2000. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Attention Deficit Hyperactivity Disorder
Source: FDA Label

METHYLIN ER Boxed Warning

ABUSE AND DEPENDENCE C N S stimulants, including methylphenidate hydrochloride extended-release capsules , other methylphenidate-containing products, and amphetamines, have a high potential for abuse and dependence. Assess the risk of abuse prior to prescribing, and monitor for signs of abuse and dependence while on therapy [see Warnings and Precautions ( 5.1 ), Drug Abuse and Dependence ( 9.2 , 9.3 )] . WARNING: ABUSE AND DEPENDENCE See full prescribing information for complete boxed warning. C...

METHYLIN ER Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

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Clinical Trial Registry

14 trials
Trial Sponsor ID Phase Status Title
NCT01628029 results posted 2012-0120 NCI-2012-01352, 2012-0120 Ph 2 active not recruiting Cognitive Behavioral Therapy and Multimodal Therapy in Treating Sleep Disturbance in Patients With Cancer
NCT05185583 77169 Ph 2 completed Methylphenidate in Childhood Apraxia of Speech
NCT06465641 KBGS_N_of_1 113883 Ph 4 recruiting Methylphenidate in KBG Syndrome: N-of-1 Series
NCT04152629 reFOQus CAN-MA-FOQ-001 Ph 4 completed Real World Evidence of the Efficacy and Safety of FOQUEST
NCT00763971 results posted SPD489-325 2008-000679-90 Ph 3 completed Randomized, Double-blind Safety and Efficacy Study of Lisdexamfetamine Dimesylate (LDX) in Children and Adolescents Aged 6-17
NCT01552902 results posted SPD489-406 2011-005452-34 Ph 4 completed Effectiveness of Vyvanse Compared to Concerta in Adolescents With Attention-deficit/Hyperactivity Disorder
NCT01183234 results posted SPD544-101 Ph 1 completed SPD544 High Strength Bioequivalence Study
NCT01552915 results posted SPD489-405 Ph 4 completed Effectiveness of Vyvanse Compared to Concerta in Adolescents With Attention-deficit/Hyperactivity Disorder
NCT02247986 140193 14-M-0193 Ph 1, Ph 2 withdrawn Investigating the Impact of Methylphenidate on Neural Response in Disruptive Behavioral Disorder
NCT01914822 275-13-RMB Ritalin version 5 Ph 2 completed The Effect Methylphenidate Hydrochloride on Pain and Auditory Sensitivity in Healthy Subjects
NCT00376675 results posted NCCTG-N05C7 NCI-2012-02701, CDR0000495148 Ph 3 completed Methylphenidate in Treating Patients With Fatigue Caused by Cancer
NCT00593853 LEUPR_L_01 07-0350-C Ph 2 terminated Efficacy Study of Methylphenidate Hydrochloride to Reduce Fatigue in Prostate Cancer Patients Receiving Hormone Therapy
NCT01348607 results posted SCUSF 0803 SCUSF-0803, 5U10CA081920-11 Ph 2 terminated Methylphenidate HCl or Modafinil in Treating Young Patients With Excessive Daytime Sleepiness After Cancer Therapy
NCT00730249 QUMEA 6520-0650-13 Ph 3 completed Quality Assurance of Administering Methylphenidate in Adults With Attention Deficit Hyperactivity Disorder (ADHD) - QUMEA
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Active Pipeline

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

METHYLIN ER FDA Label Details

Indications & Usage

METHYLIN ER is indicated for the treatment of Attention Deficit Hyperactivity Disorder.

⚠️ BOXED WARNING

WARNING: ABUSE AND DEPENDENCE C N S stimulants, including methylphenidate hydrochloride extended-release capsules , other methylphenidate-containing products, and amphetamines, have a high potential for abuse and dependence. Assess the risk of abuse prior to prescribing, and monitor for signs of abu...

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.