TheraRadar
Data updated: May 26, 2026

OCTREOTIDE ACETATE

Endocrine Approved 2005-04-08

Octreotide acetate is indicated to reduce blood levels of growth hormone (GH) and insulin growth factor-1 (IGF-1) in patients with acromegaly who have had an inadequate response to, or are not candidates for, surgical resection, pituitary irradiation, or maximally tolerated doses of bromocriptine mesylate. It is also indicated for the

Source: FDA Label • Sun Pharma

How OCTREOTIDE ACETATE Works

This medication works by mimicking the actions of the natural hormone somatostatin to inhibit the release of growth hormone, insulin, and glucagon. It also suppresses various other hormones and proteins, such as serotonin and gastrin, while decreasing blood flow to the internal organs. These combined effects help manage the symptoms caused by hormone-secreting tumors.

Source: FDA Label
15
Indications
--
Phase 3 Trials
21
Years on Market

Details

Status
Discontinued
First Approved
2005-04-08
Routes
INJECTION
Dosage Forms
INJECTABLE

OCTREOTIDE ACETATE Approval History

2006
2007
2008
2009
2010
2011
2012
2013
2014
2015
2016
2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
149 FDA actions from 2005 to 2025
Dec 2025 ORIGINAL
Update
Oct 2024 SUPPL
Label · Labeling
Sep 2024 SUPPL
Label · Labeling

What OCTREOTIDE ACETATE Treats

3 indications

OCTREOTIDE ACETATE is approved for 3 conditions since its original approval in 2005. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Acromegaly
  • Metastatic carcinoid tumors
  • Vasoactive intestinal peptide tumors (VIPomas)
Source: FDA Label

OCTREOTIDE ACETATE Competitive Set

Pro

Three rings of competition based on shared molecular targets and treated indications.

Direct competitors

2

Same target(s) AND same indication — head-to-head.

Indication competitors

4

Same indication, different mechanism — what else might this patient receive?

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to OCTREOTIDE ACETATE

3 of 10

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

BYNFEZIA PEN
OCTREOTIDE ACETATE
1 shared
Sun Pharma
Shared indications:
Acromegaly
LANREOTIDE ACETATE
LANREOTIDE ACETATE
1 shared
INVAGEN PHARMS
Shared indications:
Acromegaly
MYCAPSSA
OCTREOTIDE ACETATE
1 shared
CHIESI
Shared indications:
Acromegaly
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Clinical Trial Registry

9 trials
Trial Sponsor ID Phase Status Title
NCT03879694 I 79518 NCI-2019-00827, I 79518 Ph 1 completed Survivin Long Peptide Vaccine in Treating Patients With Metastatic Neuroendocrine Tumors
NCT06558422 AAAU9702 P30DK063608, K12DK133995 Ph 1 not yet recruiting Human Models of Selective Insulin Resistance: Pancreatic Clamp
NCT05724134 AAAU3014 3P30DK063608 Ph 1 completed Pancreatic Clamp in NAFLD
NCT06126354 AAAU7680 3P30DK063608 Ph 1 withdrawn Dexamethasone/Pancreatic Clamp P&F
NCT01229943 results posted NCI-2011-02609 NCI-2011-02609, CDR0000687459 Ph 2 completed Everolimus and Octreotide Acetate With or Without Bevacizumab in Treating Patients With Locally Advanced or Metastatic Pancreatic Neuroendocrine Tumors That Cannot Be Removed by Surgery
NCT04129255 CSMS99 IMMUNeOCT Ph 2 completed Octreotide LAR in the Induction of Immunologic Response in NENs Patients
NCT02195635 LX1606.1-109-NRM LX1606.109 Ph 1 completed Phase 1, Open-label, Drug-drug Interaction Study With Octreotide Acetate Injection and Telotristat Etiprate in Healthy Subjects
NCT01204476 NCI-2010-02196 NCI-2010-02196, CDR0000685267 Ph 1 completed Cixutumumab, Everolimus, and Octreotide Acetate in Treating Patients With Advanced Low to Intermediate Grade Neuroendocrine Carcinoma
NCT01469338 4P-11-3 NCI-2011-03266 Ph 2 terminated Cabazitaxel Plus Prednisone With Octreotide For Castration-Resistant Prostate Cancer (CRPC) Previously Treated With Docetaxel
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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

OCTREOTIDE ACETATE FDA Label Details

Indications & Usage

OCTREOTIDE ACETATE is indicated for the treatment of Acromegaly; Metastatic carcinoid tumors; Vasoactive intestinal peptide tumors (VIPomas).

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OCTREOTIDE ACETATE (PRESERVATIVE FREE)

Full clinical data, patents, trials, and competitive landscape for octreotide acetate.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.