TheraRadar
Data updated: May 26, 2026

AXUMIN (fluciclovine f-18)

Positron Emitting Activity
Oncology Approved 2016-05-27

Axumin is a radioactive diagnostic agent used for positron emission tomography (PET) imaging in men. It helps clinicians identify suspected prostate cancer recurrence in patients who show rising prostate specific antigen (PSA) levels after their initial treatment. This imaging tool allows for the visualization of potential cancer sites to assist in follow-up care.

Source: FDA Label • BLUE EARTH • Radioactive Diagnostic Agent

How AXUMIN Works

This agent works by acting as a synthetic amino acid that enters cells through specific transporters, such as LAT-1 and ASCT2. These transporters are found in higher amounts on the surface of prostate cancer cells compared to healthy tissue. As a result, the drug is taken up more heavily by cancerous cells, making them visible during a PET scan.

1
Indication
--
Phase 3 Trials
1
Priority Reviews
9
Years on Market

Details

Status
Prescription
First Approved
2016-05-27
Patent Cliff
2042

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Routes
INTRAVENOUS
Dosage Forms
SOLUTION

Companies

Active Ingredient: FLUCICLOVINE F-18

AXUMIN Approval History

2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
4 FDA actions from 2016 to 2021
May 2021 SUPPL
Label · Labeling
Jan 2017 SUPPL
Mfg · Manufacturing (CMC)
Dec 2016 SUPPL
Mfg · Manufacturing (CMC)

What AXUMIN Treats

1 indications

AXUMIN is approved for 1 conditions since its original approval in 2016. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Prostate Cancer Recurrence
Source: FDA Label

AXUMIN Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

What's emerging in AXUMIN's indications

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Phase 3 candidates targeting molecules with no FDA-approved drug, in indications AXUMIN treats. First-in-class if their pivotal trials read out positive.

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Active Pipeline

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Key Completed Trials

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

AXUMIN FDA Label Details

Indications & Usage

FDA Label (PDF)

AXUMIN is indicated for the treatment of Prostate Cancer Recurrence.

View full patent landscape →
8 OB patents · 3 families · 62 international docs across 17 countries

AXUMIN Patents & Exclusivity

Latest Patent: Apr 2042

Patents (8 active)

US11980674 Expires Apr 23, 2042
US10124079 Expires Dec 30, 2035
US10716868 Expires Dec 30, 2035
US10967077 Expires Dec 30, 2035
US10933147 Expires Dec 30, 2035
US9387266 Expires Nov 28, 2026
US10953112 Expires Nov 28, 2026
US10010632 Expires Nov 28, 2026
Source: FDA Orange Book

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Patent Timeline

  • Cliff: 2042
  • 8 active patents

Trial Analysis

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  • Development stage analysis

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.