TheraRadar
Data updated: May 26, 2026

SANCUSO (granisetron)

Serotonin 3 Receptor Antagonists
Oncology Approved 2008-09-12

Sancuso is indicated for the prevention of nausea and vomiting in adults receiving moderately or highly emetogenic chemotherapy regimens for up to five consecutive days. This transdermal system provides a prophylactic option for patients undergoing multi-day chemotherapy cycles.

Source: FDA Label • CUMBERLAND • Serotonin-3 Receptor Antagonist

How SANCUSO Works

Granisetron is a selective 5-HT3 receptor antagonist. During chemotherapy, mucosal enterochromaffin cells release serotonin, which stimulates 5-HT3 receptors located on peripheral vagal nerve terminals and centrally in the chemoreceptor trigger zone. By blocking these receptors, granisetron prevents the vagal afferent discharge and subsequent signaling that induces the vomiting reflex.

1
Indication
--
Phase 3 Trials
17
Years on Market

Details

Status
Prescription
First Approved
2008-09-12
Routes
TRANSDERMAL
Dosage Forms
FILM, EXTENDED RELEASE

Companies

Active Ingredient: GRANISETRON

SANCUSO Approval History

2009
2010
2011
2012
2013
2014
2015
2016
2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
11 FDA actions from 2008 to 2024
Sep 2024 SUPPL
Label · Labeling
Dec 2022 SUPPL
Mfg · Manufacturing (CMC)
Apr 2020 SUPPL
Label · Labeling

What SANCUSO Treats

2 indications

SANCUSO is approved for 2 conditions since its original approval in 2008. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Nausea
  • Vomiting
Source: FDA Label

SANCUSO Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

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Clinical Trial Registry

22 trials
Trial Sponsor ID Phase Status Title
NCT02858310 results posted 160154 16-C-0154 Ph 1, Ph 2 completed E7 TCR T Cells for Human Papillomavirus-Associated Cancers
NCT07401745 TMD R.25.10.27 Ph 4 active not recruiting Occlusal Splint Combined With Granisetron Injection for Management of Myofascial Pain Related to Temporomandibular Disorders
NCT07360431 GRAN-PONV-LC Ph 4 not yet recruiting Granisetron Combined With Dexamethasone or Metoclopramide for PONV Prevention After Laparoscopic Cholecystectomy
NCT03817970 18-1752.cc R01GM123330 Ph 3 active not recruiting Cisplatin Disposition and Kidney Injury
NCT00868764 392MD/40/C Ph 1 completed An Investigation on the Effect of Age and BMI on the Pharmacokinetics of Transdermal Granisetron
NCT00873197 392MD/41/C Ph 1 completed PK, Tolerability and Safety of the Co-administration of Sancuso® (Transdermal Granisetron) and IV Granisetron
NCT00890565 392MD/39/C Ph 1 completed Safety Study of Electrocardiogram (ECG) Effects of Sancuso® (Granisetron TDS)
NCT04501211 1706966663 Ph 2 withdrawn Open Label Transdermal Granisetron to Relieve Chronic Nausea and Emesis
NCT05087615 PONV ManoochehrEbrahimian Ph 3 completed Effects of Ondansetron, Metoclopramide and Granisetron on Perioperative Nausea and Vomiting in Patients Undergone Bariatric Surgery
NCT03483870 Granisetron in C.S Ph 2 completed Effect of Granisetron on Morphine Induced Pruritus in Cesarean Section
NCT04918862 MS-380-2020 Ph 3 completed A COMPARATIVE STUDY BETWEEN 1MG AND 3 MG OF GRANISETRON IN THE PREVENTION OF POSTOPERATIVE NAUSEA AND VOMITING IN STRABISMUS OPHTHALMIC SURGERIES DURING GENERAL ANESTHESIA
NCT01536392 results posted 2011-1107 NCI-2012-00221 Ph 3 completed Oral Ondansetron Versus Transdermal Granisetron (Sancuso) for Women With Cervical, Endometrial or Vaginal Cancer Receiving Pelvic Chemoradiation
NCT04613726 B.30.2.ATA.0.01.00/166 Ph 3 completed The Effect of Intravenous Granisetron and Ondansetron in Patients Undergoing Cesarean Section
NCT03503292 results posted 17-011283 Ph 4 completed Pharmacogenomics and Post-Operative Nausea and Vomiting
NCT02457195 GTPPONV results posted HRP-592 Ph 2 completed Granisetron Transdermal Patch for Prevention of Postoperative Nausea and Vomiting
NCT01183481 results posted RINV Prophylaxis Ph 2 terminated Aprepitant and Granisetron for the Prophylaxis of Radiation Induced Nausea and Vomiting - A Pilot Study
NCT02588547 SM102015 Ph 2 completed Prevention of Spinal Induced Shivering During CS
NCT00952341 results posted 0869-169 2009_626 Ph 3 completed Aprepitant/MK0869 for Prevention of Chemotherapy Induced Nausea and Vomiting Associated With Cisplatin (0869-169)(COMPLETED)
NCT01499849 results posted TS-P04832 Ph 3 completed Ph3 Safety/Efficacy Study of Rolapitant for the Prevention of CINV in Subjects Receiving Highly Emetogenic Chemotherapy
NCT01500226 results posted TS-P04834 Ph 3 completed Ph 3 Safety/Efficacy Study of Rolapitant for Prevention of CINV in Subjects Receiving Moderately Emetogenic Chemotherapy
NCT01500213 HEC results posted TS-P04833 Ph 3 completed Ph3 Safety/Efficacy Study of Rolapitant for the Prevention of CINV in Subjects Receiving Highly Emetogenic Chemotherapy
NCT01909856 sim-palonosetron Ph 2 completed The Efficacy and Safety of Palonosetron in Preventing the Gastrointestinal Reactions Induced by 3-day Highly Emetogenic Chemotherapy
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Active Pipeline

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

SANCUSO FDA Label Details

Indications & Usage

FDA Label (PDF)

SANCUSO is indicated for the treatment of Nausea; Vomiting.

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.