TheraRadar
Data updated: May 26, 2026

CYRAMZA (ramucirumab)

VEGFR2 Inhibitors Genetically Validated Trial Activity: Stable 41 active trials
Oncology Approved 2014-04-21

CYRAMZA is indicated for the treatment of Gastric Cancer; Gastroesophageal Junction Adenocarcinoma; Non-Small Cell Lung Cancer; Colorectal Cancer; Hepatocellular Carcinoma.

Source: FDA Label • Eli Lilly • Vascular Endothelial Growth Factor Receptor 2 Antagonist

How CYRAMZA Works

Ramucirumab functions by specifically binding to VEGFR2, which prevents the receptor from interacting with its ligands, including VEGF-A, VEGF-C, and VEGF-D. By blocking these interactions, the drug inhibits the ligand-stimulated activation of the receptor. This process suppresses the proliferation and migration of human endothelial cells. Ultimately, this mechanism inhibits angiogenesis, the formation of new blood vessels that support tumor growth.

Development Insights

Eli Lilly and Company conducting 39 trials (34%)
195 indications explored (Broad Platform)
gastric adenocarcinoma (14 trials)
gastroesophageal junction adenocarcinoma (14 trials)
non-small cell lung cancer (13 trials)
8
Indications
--
Phase 3 Trials
3
Priority Reviews
12
Years on Market

Details

Status
Prescription
First Approved
2014-04-21
Patent Cliff
2026
Revenue
$200M (Q4-2025)

Pro Metrics

Patent cliff and revenue data

Unlock with Pro
Routes
INJECTION
Dosage Forms
INJECTABLE

Companies

Active Ingredient: RAMUCIRUMAB

CYRAMZA Approval History

2015
2016
2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
34 FDA actions from 2014 to 2025 · 7 indication expansions
Aug 2025 SUPPL
Label · Labeling
Apr 2025 SUPPL Priority
Efficacy
Jan 2025 SUPPL
Efficacy

What CYRAMZA Treats

5 indications

CYRAMZA is approved for 5 conditions since its original approval in 2014. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Gastric Cancer
  • Gastroesophageal Junction Adenocarcinoma
  • Non-Small Cell Lung Cancer
  • Colorectal Cancer
  • Hepatocellular Carcinoma
Source: FDA Label

CYRAMZA Target & Pathway

Pro

Target

VEGFR (Vascular Endothelial Growth Factor Receptor) Growth Factor Receptor

Receptors on blood vessel cells that respond to VEGF signals to form new blood vessels. Cancer cells exploit this pathway to ensure blood supply for tumor growth. Blocking VEGFRs prevents tumor angiogenesis and limits cancer progression.

Pathway Context

VEGFR on blood vessels is activated by VEGF to promote angiogenesis

VEGF (Vascular Endothelial Growth Factor) ligand

A signaling protein that stimulates the formation of new blood vessels (angiogenesis). Tumors need blood supply to grow, so they secrete VEGF to create new vessels. Blocking VEGF starves tumors of oxygen and nutrients, inhibiting their growth.

CYRAMZA Competitive Set

Pro

Three rings of competition based on shared molecular targets and treated indications.

Unlock 11 more competitors across all three rings.
Upgrade to Pro

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to CYRAMZA

3 of 20

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

KEYTRUDA
PEMBROLIZUMAB
4 shared
Merck
Shared indications:
Non-Small Cell Lung CancerGastric CancerHepatocellular Carcinoma +1 more
OPDIVO
NIVOLUMAB
4 shared
Bristol-Myers Squibb
Shared indications:
Non-Small Cell Lung CancerColorectal CancerHepatocellular Carcinoma +1 more
CAPECITABINE
CAPECITABINE
2 shared
AMNEAL PHARMS
Shared indications:
Colorectal CancerGastric Cancer
📋

Clinical Trial Registry

115 trials
Trial Sponsor ID Phase Status Title
NCT04310007 NCI-2020-01541 NCI-2020-01541, EA5191 Ph 2 active not recruiting Testing the Addition of the Pill Chemotherapy, Cabozantinib, to the Standard Immune Therapy Nivolumab Compared to Standard Chemotherapy for Non-small Cell Lung Cancer
NCT04704934 DS8201-A-U306 2020-004559-34 Ph 3 active not recruiting Trastuzumab Deruxtecan for Subjects With HER2-Positive Gastric Cancer or Gastro-Esophageal Junction Adenocarcinoma After Progression on or After a Trastuzumab-Containing Regimen (DESTINY-Gastric04)
NCT06203600 NCI-2023-11064 NCI-2023-11064, S2303 Ph 2, Ph 3 recruiting Adding Nivolumab to Usual Treatment for People With Advanced Stomach or Esophageal Cancer, PARAMUNE Trial
NCT06448754 eVOLVE-01 D798KC00001 2023-509482-20-00 Ph 2 recruiting Volrustomig Priming Regimens Exploratory Phase II Platform Study
NCT06445972 3475-06D 2023-509306-29-00, U1111-1299-8160 Ph 1, Ph 2 recruiting Substudy 06D: Combination Therapies in Second Line (2L) Gastroesophageal Adenocarcinoma (MK-3475-06D/Keymaker-U06)
NCT06043427 GA4 Ph 2 recruiting Paclitaxel and Ramucirumab +/- Zanidatamab in HER2 Postive Advanced Gastroesophageal Adenocarcinoma
NCT04145349 results posted 17305 J1S-MC-JV01, 2018-004242-42 Ph 1, Ph 2 completed CAMPFIRE: A Study of Ramucirumab (LY3009806) in Children and Young Adults With Desmoplastic Small Round Cell Tumor
NCT05642572 S1900G NCI-2022-09254, S1900G Ph 2 recruiting Comparing Combinations of Targeted Drugs for Advanced Non-Small Cell Lung Cancer That Has EGFR and MET Gene Changes (A Lung-MAP Treatment Trial)
NCT05365581 2138-CL-0101 jRCT2031210644, CTR20241945 Ph 1 recruiting A Study of ASP2138 Given by Itself or Given With Other Cancer Treatments in Adults With Stomach Cancer, Gastroesophageal Junction Cancer, or Pancreatic Cancer
NCT06616584 S1800E NCI-2024-06444, S1800E Ph 2, Ph 3 recruiting Adding the Immunotherapy Drug Cemiplimab to Usual Treatment for People With Advanced Non-Small Cell Lung Cancer Who Had Previous Treatment With Platinum Chemotherapy and Immunotherapy (An Expanded Lung-MAP Treatment Trial)
NCT06031688 S1900K NCI-2023-04727, S1900K Ph 2 recruiting Targeted Treatment for Advanced Non-Small Cell Lung Cancer That Has a MET Exon 14 Skipping Gene Change (An Expanded Lung-MAP Treatment Trial)
NCT03650764 201809094 Ph 1, Ph 2 completed Ramucirumab + Pembrolizumab in Patients With Recurrent/Metastatic Head and Neck Squamous Cell Carcinoma
NCT06996782 ALTAIR D702KC00001 2024-519786-22 Ph 1, Ph 2 recruiting A Platform Study in Non-Small Cell Lung Cancer (NSCLC)
NCT07098338 LIBRA D6187C00001 Ph 2 recruiting A Study of Novel Combinations in Non-Small Cell Lung Cancer (NSCLC)
NCT07546812 GS-US-742-7757 2025-524095-27 Ph 2 recruiting Study of Denikitug (GS-1811) Given Alone or With Nivolumab or Chemotherapy in Adults With Metastatic Gastric, Gastroesophageal Junction (GEJ), and Esophageal Adenocarcinomas
NCT03909334 HCRN LUN18-335 Ph 2 active not recruiting Study of Osimertinib With and Without Ramucirumab in Locally Advanced or Metastatic Non-Small Cell Lung Cancer (NSCLC)
NCT05633602 S2302 NCI-2022-09319, S2302 Ph 3 active not recruiting Ramucirumab Plus Pembrolizumab vs Usual Care for Treatment of Stage IV or Recurrent Non-Small Cell Lung Cancer Following Immunotherapy, Pragmatica-Lung Study
NCT03081143 RAMIRIS RAMIRIS AIO-STO-0415 Ph 2, Ph 3 active not recruiting Ramucirumab Plus FOLFIRI Versus Ramucirumab Plus Paclitaxel in Patients With Advanced or Metastatic Gastric Cancer, Who Failed One Prior Line of Palliative Chemotherapy
NCT06007937 23-131 Ph 1, Ph 2 recruiting A Study of Lorlatinib in Combination With Ramucirumab in People With Lung Cancer
NCT03798626 CVPM087A2101 2018-003952-19 Ph 1 completed Gevokizumab With Standard of Care Anti-cancer Therapies for Metastatic Colorectal, Gastroesophageal, and Renal Cancers
NCT05980000 Rambro2 202308161 Ph 2 active not recruiting Ramucirumab and Pembrolizumab vs Pembrolizumab Monotherapy in PD-L1 Positive Head and Neck Squamous-Cell Carcinoma
NCT05999994 CAMPFIRE 17304 J1S-MC-JAAA Ph 2 recruiting A Master Protocol (LY900023) That Includes Several Clinical Trials of Drugs for Children and Young Adults With Cancer
NCT04921904 020-055 Ph 1, Ph 2 active not recruiting Abemaciclib Plus Ramucirumab for Esophageal/Gastroesophageal Junction Ca
NCT06771622 HCB101-201 Ph 1, Ph 2 active not recruiting Safety and Efficacy of HCB101 in Combination With Multiple Agents in Patients With Advanced Solid Tumors
NCT03008278 results posted NCI-2016-02049 NCI-2016-02049, 2000021407 Ph 1, Ph 2 completed Olaparib and Ramucirumab in Treating Patients With Metastatic or Locally Recurrent Gastric or Gastroesophageal Junction Cancer That Cannot Be Removed by Surgery
NCT04340882 DoceRamPem STUDY00000030 NCI-2020-01134, WINSHIP4950-20 Ph 2 active not recruiting Phase 2 DoceRamPem for Patients With Metastatic or Recurrent NSCLC Who Progressed on Platinum-Doublet and PD-1/PD-L1 Blockade
NCT02411448 RELAY results posted 15540 I4T-MC-JVCY, 2014-004824-22 Ph 3 active not recruiting A Study of Ramucirumab (LY3009806) in Combination With Erlotinib in Previously Untreated Participants With EGFR Mutation-Positive Metastatic NSCLC (RELAY)
NCT03527108 TH-189 TH-189 Ph 2 active not recruiting Nivolumab Plus Ramucirumab in Patients With Recurrent, Advanced, Metastatic NSCLC
NCT04332367 UPCC 05519 IRB833759 Ph 2 recruiting Carboplatin, Taxane And Ramucirumab for Patients With NSCLC After Pemetrexed or Pembrolizumab Maintenance
NCT03281369 YO39609 2016-004529-17 Ph 1, Ph 2 completed A Study of Multiple Immunotherapy-Based Treatment Combinations in Patients With Locally Advanced Unresectable or Metastatic Gastric or Gastroesophageal Junction Cancer (G/GEJ) or Esophageal Cancer (Morpheus-Gastric and Esophageal Cancer)
NCT06251973 23-361 Ph 2 active not recruiting A Study of agenT-797 in Combination With Botensilimab, Balstilimab, Ramucirumab, and Paclitaxel for People With Esophageal, Gastric, or Gastro-esophageal Junction Cancer
NCT06675136 24445 NCI-2024-08883, 24445 Ph 1 recruiting Nab-Paclitaxel PIPAC in Combination With Paclitaxel and Ramucirumab for the Treatment of Stomach Cancer With Peritoneal Metastases
NCT04205968 S1922 NCI-2019-04213, S1922 Ph 2 recruiting Ramucirumab and Paclitaxel or FOLFIRI in Advanced Small Bowel Cancers
NCT03694002 results posted S1701 NCI-2017-02254, S1701 Ph 2 completed Carboplatin and Paclitaxel With or Without Ramucirumab in Treating Patients With Locally Advanced, Recurrent, or Metastatic Thymic Cancer That Cannot Be Removed by Surgery
NCT02597036 results posted 15580 I7W-MC-JQBA, 2015-001204-64 Ph 1 terminated A Study of LY3127804 With Ramucirumab in Participants With Advanced Solid Tumors
NCT05002127 AT148006 Ph 2, Ph 3 active not recruiting A Study of Evorpacept (ALX148) in Patients With Advanced HER2+ Gastric Cancer (ASPEN-06)
NCT06038578 950GCV01 Ph 2 recruiting A Study of TRK-950 When Used in Combination With Ramucirumab and Paclitaxel in Patients With Gastric Cancer
NCT02711553 results posted 16329 I3O-MC-JSBF, 2015-004699-31 Ph 2 active not recruiting A Study of Ramucirumab (LY3009806) or Merestinib (LY2801653) in Advanced or Metastatic Biliary Tract Cancer
NCT03872947 950P1V02 Ph 1 active not recruiting A Study of TRK-950 in Combinations With Anti-Cancer Treatment Regimens in Patients With Advanced Solid Tumors
NCT04069273 SEQUEL HCRN GI18-333 Ph 2 recruiting Novel SEQUEnced Immunotherapy With Anti-angiogenesis and Chemotherapy in Advanced gastroesophageaL Adenocarcinoma
NCT04120454 results posted OSU-19132 NCI-2019-05348 Ph 2 completed Ramucirumab and Pembrolizumab for the Treatment of EGFR Mutant Recurrent or Metastatic Non-small Cell Lung Cancer
NCT02678182 PLATFORM 3804 Ph 2 active not recruiting Planning Treatment for Oesophago-gastric Cancer: a Maintenance Therapy Trial
NCT04394624 CARMEN-LC04 results posted ACT16525 U1111-1244-1585, 2019-003914-15 Ph 2 terminated Tusamitamab Ravtansine (SAR408701) in Combination With Ramucirumab or Ramucirumab and Pembrolizumab in Pretreated Patients With NSQ NSCLC (CARMEN-LC04)
NCT05096663 S1800D NCI-2021-09852, S1800D Ph 2, Ph 3 active not recruiting Testing the Use of Combination Immunotherapy Treatment (N-803 [ALT-803] Plus Pembrolizumab) Against the Usual Treatment for Advanced Non-small Cell Lung Cancer (A Lung-MAP Treatment Trial)
NCT03560973 RAMES GOIRC-03-2016 Ph 2 completed A Double Blind, Placebo Controlled, Randomized Phase II Study Evaluating Gemcitabine With or Without Ramucirumab , for II Line Treatment MPM
NCT05062980 Acclaim-2 ONC-004 Ph 1, Ph 2 terminated Quaratusugene Ozeplasmid (Reqorsa) in Combination With Pembrolizumab in Previously Treated Non-Small Lung Cancer
NCT02795858 results posted 16-072 Ph 2 completed A Phase II Study of Ramucirumab With Somatostatin Analog Therapy in Patients With Advanced, Progressive Carcinoid Tumors
NCT04499924 MOUNTAINEER-02 results posted SGNTUC-022 C4251004 Ph 2, Ph 3 completed Tucatinib, Trastuzumab, Ramucirumab, and Paclitaxel Versus Paclitaxel and Ramucirumab in Previously Treated HER2+ Gastroesophageal Cancer
NCT02581215 results posted HCRN GI14-198 Ph 2 completed Phase II Randomized Trial of mFOLFIRINOX +/- Ramucirumab in Advanced Pancreatic Cancer
NCT02791334 PACT 16088 I8J-MC-JYCA, 2016-000440-33 Ph 1 completed A Study of Anti-PD-L1 Checkpoint Antibody (LY3300054) Alone and in Combination in Participants With Advanced Refractory Solid Tumors

Showing 50 of 115 trials

🔬

Active Pipeline

Pro

Ongoing clinical trials by development phase

Loading...

Key Completed Trials

Pro

Completed studies with published results, ranked by significance

Loading...
📊

Trial Timeline

Full development history with FDA approval milestones

|
Loading...
Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

CYRAMZA FDA Label Details

Indications & Usage

FDA Label (PDF)

CYRAMZA is indicated for the treatment of Gastric Cancer; Gastroesophageal Junction Adenocarcinoma; Non-Small Cell Lung Cancer; Colorectal Cancer; Hepatocellular Carcinoma.

Pro Intelligence Preview

Deep insights for CYRAMZA

Revenue Insights

  • Q4-2025: $200M
  • Historical trend analysis

Patent Timeline

  • Cliff: 2026
  • Generic/biosimilar risk

Trial Analysis

  • 114 total trials
  • Stage: Stable

Competitive Landscape

  • 20 similar drugs
  • Same target/indication analysis
Unlock Full Intelligence

Full approval history • All patents • Revenue trends • Competitor analysis

Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment