TheraRadar
Data updated: May 26, 2026

ZTALMY (ganaxolone)

GABA A Receptor Positive Modulators Trial Activity: Declining 1 active trials
First-in-Class Priority Review
CNS Approved 2022-03-18

ZTALMY is indicated for the treatment of Seizures; Cyclin-Dependent Kinase-Like 5 Deficiency Disorder.

Source: FDA Label • IMMEDICA PHARMA • Neuroactive Steroid Gamma-Aminobutyric Acid A Receptor Positive Modulator

How ZTALMY Works

While the precise mechanism of ganaxolone is unknown, its therapeutic effects are thought to result from its activity in the central nervous system. The drug acts as a positive allosteric modulator of the gamma-aminobutyric acid type A (GABA A) receptor. By modulating these receptors, the medication produces anticonvulsant effects to help manage seizures.

Development Insights

Marinus Pharmaceuticals conducting 15 trials (88%)
25 indications explored (Broad Platform)
cdkl5 deficiency disorder (2 trials)
tuberous sclerosis complex (2 trials)
depressive disorder (2 trials)
2
Indications
--
Phase 3 Trials
1
Priority Reviews
4
Years on Market

Details

Status
Prescription
First Approved
2022-03-18
Patent Cliff
2042

Pro Metrics

Patent cliff and revenue data

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Routes
ORAL
Dosage Forms
SUSPENSION

Companies

Active Ingredient: GANAXOLONE

ZTALMY Approval History

2023
2024
2025
2026
Original
New Indication
New Form
Label Update
8 FDA actions from 2022 to 2025
Oct 2025 SUPPL
Label · Labeling
Aug 2025 SUPPL
Label · Labeling
Jun 2023 SUPPL
Label · Labeling

What ZTALMY Treats

2 indications

ZTALMY is approved for 2 conditions since its original approval in 2022. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Seizures
  • Cyclin-Dependent Kinase-Like 5 Deficiency Disorder
Source: FDA Label

ZTALMY Competitive Set

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Three rings of competition based on shared molecular targets and treated indications.

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to ZTALMY

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Clinical Trial Registry

17 trials
Trial Sponsor ID Phase Status Title
NCT05249556 1042-CDD-3002 Ph 3 not yet recruiting Double-blind, Randomized, Placebo-controlled Trial of Ganaxolone in CDKL5 Deficiency Patients 6 Months to Less Than 2 Years Old
NCT05604170 results posted 1042-TSC-3002 Ph 3 terminated Open-label Study of Adjunctive GNX Treatment in Children and Adults With TSC-related Epilepsy
NCT05323734 results posted 1042-TSC-3001 Ph 3 completed Adjunctive GNX Treatment Compared With Placebo in Children and Adults With TSC-related Epilepsy
NCT04391569 RAISE results posted 1042-SE-3003 Ph 3 completed Randomized Therapy In Status Epilepticus
NCT05814523 1042-SE-3004 Ph 3 withdrawn To Evaluate the Efficacy, Safety, and Tolerability of Intravenous Ganaxolone Added to Standard of Care in Refractory Status Epilepticus (RSE)
NCT03460756 results posted 1042-PPD-2003 Ph 2 completed A Clinical Trial of Oral Ganaxolone in Women With Postpartum Depression
NCT03228394 results posted 1042-PPD-2002 Ph 2 completed A Clinical Trial of Intravenous (IV) Ganaxolone in Women With Postpartum Depression
NCT02519439 results posted 1042-0604 Ph 3 terminated A Two-year Open-label Extension Study of Ganaxolone in Patients With Drug-resistant Partial-onset Seizures
NCT03865732 results posted 1042-PCDH19-3002 2018-004496-12 Ph 2 completed Study of Adjunctive Ganaxolone Treatment in Female Children With Protocadherin 19 (PCDH19)-Related Epilepsy (Violet Study)
NCT03572933 Marigold results posted 1042-CDD-3001 2018-001180-23 Ph 3 completed Study of Adjunctive Ganaxolone Treatment in Children and Young Adults With CDKL5 Deficiency Disorder
NCT01725152 results posted 1042-0800 Ph 2 completed Ganaxolone Treatment in Children With Fragile X Syndrome
NCT04285346 TSC results posted 1042-TSC-2001 Ph 2 completed Adjunctive Ganaxolone Treatment (Part A) in TSC Followed by Long-term Treatment (Part B)
NCT02358538 results posted 1042-900 Ph 2 completed Open-Label PoC Trial of Ganaxolone in Children With PCDH19 Female Pediatric Epilepsy and Other Rare Genetic Epilepsies
NCT01963208 results posted 1042-0603 Ph 3 completed Phase 3 Study of Adjunctive Ganaxolone in Adults With Drug-resistant Partial Onset Seizures and Open-label Extension
NCT01339689 results posted 1042-0700 Ph 2 completed Ganaxolone in Posttraumatic Stress Disorder (PTSD)
NCT01002820 0602 results posted 1042-0602 Ph 2 completed A Treatment Use Protocol for Subjects Continuing on From the Open-label Extension 0601
NCT01857531 Ganaxolone results posted Pro00041533 1P50DA027840-01A1 Ph 2 completed Proof-Of-Concept Investigation With a Neurosteroid Analog (Ganaxolone) as a Smoking Cessation Candidate
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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

ZTALMY FDA Label Details

Indications & Usage

FDA Label (PDF)

ZTALMY is indicated for the treatment of Seizures; Cyclin-Dependent Kinase-Like 5 Deficiency Disorder.

View full patent landscape →
11 OB patents · 3 families · 116 international docs across 17 countries

ZTALMY Patents & Exclusivity

Latest Patent: Sep 2042
Exclusivity: Jun 2029

Patents (11 active)

US12115169 Expires Sep 30, 2042
US12268696 Expires Sep 30, 2042
US12144801 Expires Aug 10, 2037
US10603308 Expires Aug 10, 2037
US8318714 Expires Nov 28, 2031
US8618087 Expires Nov 28, 2026
US9056116 Expires Nov 28, 2026
US7858609 Expires Nov 28, 2026
US8022054 Expires Nov 28, 2026
US8367651 Expires Nov 28, 2026
US9029355 Expires Nov 28, 2026

Exclusivity

D-197 Until Oct 2028
NCE Until Jun 2027
ODE-395 Until Jun 2029
Source: FDA Orange Book

Pro Intelligence Preview

Deep insights for ZTALMY

Revenue Insights

  • Quarterly revenue tracking
  • Historical trend analysis

Patent Timeline

  • Cliff: 2042
  • 11 active patents

Trial Analysis

  • 17 total trials
  • Stage: Declining

Competitive Landscape

  • 20 similar drugs
  • Same target/indication analysis
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Full approval history • All patents • Revenue trends • Competitor analysis

Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.

How We Calculate These Metrics

Trial Activity Stage

Measures the current development activity pattern based on trial phases, status, and trends. Important: This measures R&D activity, not commercial lifecycle.

Trial statuses: "Active" means recruiting or ongoing. "Completed" means reached planned endpoint. "Terminated" means stopped early—often due to safety, efficacy, or business reasons.

  • Growth: High proportion of early-phase trials (Phase 1/2), active development
  • Expansion: Significant Phase 3 activity, approaching or pursuing approvals
  • Mature: Substantial Phase 4 post-marketing studies
  • Stable: Mixed phase distribution, steady development
  • Declining: Low active trial ratio, reduced R&D investment