TheraRadar
Data updated: May 26, 2026

LOCAMETZ (gallium ga-68 gozetotide)

Oncology Approved 2022-03-23

Locametz is a radioactive diagnostic agent used during PET scans to identify prostate-specific membrane antigen (PSMA)-positive lesions in men with prostate cancer. It helps clinicians evaluate patients with suspected metastasis before they begin initial therapy or those with rising PSA levels that suggest the cancer has returned. Additionally, this tool helps identify which patients are suitable candidates for targeted PSMA-directed therapies.

Source: FDA Label • Novartis

How LOCAMETZ Works

This agent works by binding to PSMA, a protein frequently found in high amounts on the surface of malignant prostate cancer cells. Because it contains gallium-68, a radionuclide that emits positrons, it allows for the visualization of these cancer cells through PET imaging.

1
Indication
--
Phase 3 Trials
4
Years on Market

Details

Status
Prescription
First Approved
2022-03-23
Patent Cliff
2036

Pro Metrics

Patent cliff and revenue data

Unlock with Pro
Routes
INTRAVENOUS
Dosage Forms
POWDER

Companies

Active Ingredient: GALLIUM GA-68 GOZETOTIDE

LOCAMETZ Approval History

2023
2024
2025
2026
Original
New Indication
New Form
Label Update
2 FDA actions from 2022 to 2025
Mar 2025 SUPPL
Label · Labeling
Mar 2022 ORIGINAL
New Ingredient · Type 2 - New Active Ingredient

What LOCAMETZ Treats

3 indications

LOCAMETZ is approved for 3 conditions since its original approval in 2022. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Prostate Cancer
  • Metastasis
  • Recurrence
Source: FDA Label

LOCAMETZ Competitive Set

Pro

Three rings of competition based on shared molecular targets and treated indications.

Unlock 9 more competitors across all three rings.
Upgrade to Pro

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

What's emerging in LOCAMETZ's indications

See all emerging drugs →

Phase 3 candidates targeting molecules with no FDA-approved drug, in indications LOCAMETZ treats. First-in-class if their pivotal trials read out positive.

Drugs Similar to LOCAMETZ

3 of 20

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

GALLIUM GA-68 GOZETOTIDE
GALLIUM GA-68 GOZETOTIDE
3 shared
IONETIX
Shared indications:
Prostate CancerMetastasisRecurrence
GOZELLIX
GALLIUM GA-68 GOZETOTIDE
3 shared
TELIX INNOVATIONS
Shared indications:
Prostate CancerMetastasisRecurrence
ILLUCCIX
GALLIUM GA-68 GOZETOTIDE
3 shared
TELIX
Shared indications:
Prostate CancerMetastasisRecurrence
🔬

Active Pipeline

Pro

Ongoing clinical trials by development phase

Loading...

Key Completed Trials

Pro

Completed studies with published results, ranked by significance

Loading...
📊

Trial Timeline

Full development history with FDA approval milestones

|
Loading...
Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

LOCAMETZ FDA Label Details

Indications & Usage

FDA Label (PDF)

LOCAMETZ is indicated for the treatment of Prostate Cancer; Metastasis; Recurrence.

View full patent landscape →
2 OB patents · 2 families · 124 international docs across 17 countries

LOCAMETZ Patents & Exclusivity

Latest Patent: Mar 2036

Patents (2 active)

US12109277 Expires Mar 9, 2036
US11369590 Expires Aug 15, 2028
Source: FDA Orange Book

Pro Intelligence Preview

Deep insights for LOCAMETZ

Revenue Insights

  • Quarterly revenue tracking
  • Historical trend analysis

Patent Timeline

  • Cliff: 2036
  • 2 active patents

Trial Analysis

  • Clinical trial tracking
  • Development stage analysis

Competitive Landscape

  • 20 similar drugs
  • Same target/indication analysis
Unlock Full Intelligence

Full approval history • All patents • Revenue trends • Competitor analysis

Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.